Synthesis of DSPE-PEG-Angiopep-2To synthesize DEPE-PEG-Angiopep-2, 5 mg of DSPE-PEG-Mal was completely dissolved in 10 mL of water. Then, 6 mg of Angiopep-2-cys was added to the solution, and the mixture was stirred at 37°C for 12 hours. The solution was dialyzed (MW3500) to remove excess Angiopep-2-cys. The resulting purified product, DSPE-PEG-Angiopep-2, was then freeze-dried and stored at −20°C for subsequent usage.

DSPE-PEG-Angiopep-2的合出为了能获得DEPE-PEG-Angiopep-2,将5mg DSPE-PEG-Mal全溶水在10mL自来水中。第二步,向盐饱和溶液内加入6mg Angiopep-2-cys,并将融合物在37°C下搅伴12一小时。将盐饱和溶液透析(MW3500)以清除已有的Angiopep-2-cys。第二步将所得的纯化物品DSPE-PEG-Angiopep-2冷冻熟食太干并贮藏在-20°C下,以备前因后果便用。CG/SN-38微米微粒(NP)的制作与开始之前新闻稿件的不同,但要经过了获取。G和1 mg SN-38溶解性在20μL DMSO中,随后向水盐溶液里加入1 mL水,随后彩超清洗清洗工作分之五钟。将盐溶液剂用蒸溜水(1L)透析(MW3500)127分钟。随后,将NP水盐溶液与肯一定的巨噬癌内部彩超清洗清洗2半个7分钟,以获取巨噬癌内部/IGC/SN-38(M-NP)。不仅如此,按照彩超清洗清洗工作(400 W,2 s开/3 s关,2 min)M-NP和优先制作的100μg DSPE-PEG-Angiopep-2,获取1 mL Angiopep-2绘制的M-NP(AM-NP)。对应推见:FITC-iRGD-PEG-DSPER8-PEG-DSPEAngiopep-2-PEG-DSPEFITC-Angiopep-2-PEG-DSPETH-PEG-DSPER6H4-PEG-DSPEMPG-PEG-DSPEGE11-PEG-DSPEPTP-PEG-DSPESP94-PEG-DSPE不低于文章信息内容信息内容来源于各大刊物或学术论文,深表歉意侵权行为请电话联系人们册除!